ICM 2021 | Macao, China
★ Scientific Programme

Stage 1: Keynote Forum
-Strategic Thinkers for Next Generation Medichem

Part 1: Opening Ceremony Part 3: Master Dialogs of GALATECH
Part 2: GALATECH Plenary Summit
• Speech from WHO
• Speech from Health Ministrial Officers
• Speech from Those Entrepreneur Leaders Changing the World Health Status
• Speech from Top 10 World Class University President
• Speech from Top Healthcare Industries
• Speech from Top Biotech Industries
• Speech from Global Prize Laureates
Part 4: Keynote Forum of ICM-2021 • Disruptive Technologies in Medichem
• Emerging Drug Targets Discovery
• New Drug Chemical Modalities Discovery
• Smart Drug Design
• Preclinical Process
• Next Generation Drug Pipeline
• Integrative Discovery Chemistry Services

Stage 2: New Era of Medichem Methodology Disruptions
-Strategic Innovators Enable Early Drug Discovery

Xlab 01: AI in Medicinal Chemistry Xlab 09: Navigating Chemical and Druggable Space
Xlab 02: Big Data and ML/DL for Discovery Chemistry Xlab 10: DNA-Encoded Library (DEL) Technology
Xlab 03: VR/AR/MR for Drug Design Xlab 11: Chemical Discovery in the Era of Metabolomics
Xlab 04: Predictive Medicinal Chemistry Xlab 12: Enzyme Direct Evolution and Biotransformations in Medichem
Xlab 05: Internet of Chemistry in Drug Discovery Xlab 13: New Approaches to Drug Candidate Optimization and Characterization
Xlab 06: Robotics and Automations in Medicinal Chemistry Xlab 14: Emerging Medichem in silico
Xlab 07: CRISPR/Cas9 and Genome Editing Xlab 15: Generative Recurrent Networks for De Novo Drug Design
Xlab 08: Virtual Hit-to-Lead Optimization Xlab 16: Cheminformatics and Bioinformatics in Medichem

Stage 3: Pioneerscape of Target Druggability
-Leadership in Discovering Validated Targets

Theme 1: Targets Validation and Discovery

Family 1-1: New Strategies and Platforms for Evaluating New Drug Targets Family 1-6: Cell Biology Methods in Target Validation
Family 1-2: Reverse Translation to Support Efficient Drug Target Selection and Stratified Medicine Family 1-7: Chemical Proteomic Approach for Kinase Inhibitor Selectivity Profiling and Target Discovery
Family 1-3: Affinity-Based Chemoproteomics for Target Identification Family 1-8: Genetic Manipulation/Modulation for Target Discovery and Validation
Family 1-4: Elucidating Target Biology and Drug Mechanism of Action Across Human Cell-Based Model Systems Family 1-9: Label-Free Techniques for Target Discovery and Validation
Family 1-5: Activity-Based Protein Profiling Family 1-10: Bioinformatic Approaches in the Understanding of Mechanism of Action

Theme 2: Targeting DNA/Gene, RNA and Nuclear Receptors

Family 2-1: CRISPR/Cas9 & Targeted Genome Editing Family 2-4: Targeting Oligonucleotides
Family 2-2: Targeting miRNA,siRNA and other ncRNA Family 2-5: Epigenetic Targets
Family 2-3: Targeting DNA/Gene and DNA-DNA Interactions Family 2-6: Targeting Nuclear Receptors

Theme 3: Targeting Proteins, Emerging Receptors and Enzymes

Family 3-1: Targeting the Unfolded Protein Response Family 3-5: Targeting Membrane Protein
Family 3-2: Challenging Kinases and Phosphatase
-PI3K, PTP, SHP-2, PTP2C, PSTPS, PP2A and PP2B
Family 3-6: Targeting Histone Methyltransferases
Family 3-3: Disordered Proteins as Drug Targets Family 3-7: Targeting Emerging Receptors
Family 3-4: Targeting Metabolic Enzyme Family 3-8: Targeting CDC25 Phosphatases

Theme 4: Targeting Protein-Protein Interactions (PPIs) and Protein-DNA Interactions

Family 4-1: Advances in Targeting PPIs Family 4-4: PPI Inhibitors
Family 4-2: PPI Modeling and Drug Screening Family 4-5: Targeting Protein-Nucleic Acid Complexes
Family 4-3: PPI Modulators/Regulators Family 4-6: Science and Tech in Exploring PPI

Theme 5: Targeting Protein Degradation and PROTAC

Family 5-1: Small Molecule Degraders Family 5-6: Target the Autophagy/Lysosome Pathway
Family 5-2: Novel PROTACs Design Family 5-7: ‘Molecular glue’ Degrader
Family 5-3: Druggable Proteome Family 5-8: Genetic Fusion Strategies of Degradation Tags For Targeted Protein Degradation and The dTAG system
Family 5-4 Novel Ligases & Chaperones for Degradation Family 5-9: Macromolecular conjugates as Protein Degrader
Family 5-5: Bifunctional Degrader Family 5-10: Protein Degradation Discovery Toolbox

Theme 6: Targeting GPCR and Ion Channels

Family 6-1: GPCR-Allosteric Modulation Family 6-5: GPCR Signaling Complexities
Family 6-2: Non-Classical Signaling Family 6-7: Biased GPCR Signaling
Family 6-3: Engaging GPCRs Family 6-6: Emerging Technologies for Targeting, Assaying and Modulating Ion Channel Targets
Family 6-4: Opioid Receptors Family 6-8: Ion Channels as Therapeutic Antibody Targets

Theme 7: Druggable IO Targets

Family 7-1: Frontier of IO Targets Family 7-4: Targeted IO Therapies
Family 7-2: Immunomodulator Targets Family 7-5: Oncolytic Virus Targets in IO
Family 7-3: Cancer Vaccine Targets Family 7-6: IO Cell Therapy and Bispecific Antibody Targets

Theme 8: Drugging Undruggable Targets
-Meet the Challenges in Difficult Targets

Family 8-1: Drugging Undruggable Molecular Cancer Targets Family 8-4: RAS and KRAS
Family 8-2: Drugging “Undruggable” Genes Family 8-5: Targeting Resistant Targets
Family 8-3: Transcription factors (TFs) Family 8-6: Other Challenging Targets for Drug Design

Theme 9: Next Wave of Epigenetic-Targeting Drug Discovery
-New Dreamland of Medicinal Chemists

Family 9-1: Selecting Ideal Epi-Targets for Hackling Family 9-5: Preclinical In-Vivo Biology of Epi-drugs
Family 9-2: Epi-Biomarker Discovery Family 9-6: Advanced Tools
-New Challenges from Crispr and Genome Editing
Family 9-3: Epi-Drug Design and Synthesis Family 9-7: Pharmacology of Epi-drugs
Family 9-4: Enzymatic Assay and In Vitro Studies of Epi-Drugs Family 9-8: Clinical Trials of Epi-drugs

Theme 10: Targeting Microbiota
-New Frontier of System Chemical Biology

Family 10-1: Microbiome and Microbiota Science Family 10-5: Microbiome Discovery Goes Small Molecules
Family 10-2: The Microbiome Drug Discovery Family 10-6: Microbiome Metabolite Mimics
Family 10-3: Microbiome as a Target for Cancer Therapy Family 10-7: Microbiota Toxin and Anti-Toxin Development
Family 10-4: Advanced Microbiome Biotech Family 10-8: Microbiome Drug Clinical Trials

Stage 4: New Shapers of Drug Chemical Modalities
-Booming Achievements in Discovery New Chemical Diversities

Art Show 01: Oligonucleotides, ASOs & RNAi Art Show 07: Peptibody
Art Show 02: Next generation Peptides and Peptidomimetics Art Show 08: Protein Degraders
Art Show 03: Current Mixed Drug Modalities Art Show 09: Targeted Covalent Inhibitors (TCIs)
Art Show 04: Small Molecule-Drug Conjugates (SMDCs) Art Show 10: Fusion Protein and BiTE® Antibody Construct
Art Show 05: Molecular Conjugates for Targeted Delivery Art Show 11: Chemical Probes for Characterizing Biology
Art Show 06: RNAi, miRNA-Based Modality Therapeutics Art Show 12: Bioimaging

Stage 5: Drug Design Artists
-Intelligent Creation of Potential Hit to Leads

Art Show 01: Fragment Based Drug Design Art Show 10: In Vivo Imaging in Drug Design
Art Show 02: Structure/Biostructure-based and ligand-based drug Design Art Show 11: Systems Biology in Drug Design
-From Drug-Target Space (off-target), Systems Biology Space to Phenotype Space
Art Show 03: Novel Approaches in Silico Drug Design Art Show 12: New Chiral Drug Design
Art Show 04: Ligand-Based Drug Design Art Show 13: Multi-Target Drug Design
Art Show 05: Design based on Drug-Like Properties and Decision Making Art Show 14: Rational Receptors-based Drug Design
Art Show 06: Chemical Biology and Structural Biology in Drug Design Art Show 15: Design of an Effective Natural-Products-Based Approach
Art Show 07: Design of Hybrid Molecules Art Show 16: Prodrug-based Drug Design and Development
Art Show 08: Macrocycles in Drug Design Art Show 17: Mechanism and Pathway based Drug Design
Art Show 09: Design Long Lasting, Oral Bioavailability and Brain Penetration Art Show 18: Selective Optimization of Side Activities (SOSA) in Drug Discovery

Stage 6: Masters of New Discovery Synthetic Toolbox
-Robust Chemistry toward Desired Candidates

SynTech 01: Molecular Conjugates for Targeted Delivery SynTech 14: Chemistry of Biomarkers
SynTech 02: Discovery Click Chemistry for Drug Conjugates SynTech 15: TCM and Natural Products Drug Chemistry
SynTech 03: Antibody-Recruiting Small Molecules Constructs as Immunotherapeutics SynTech 16: Biomaterial/Biopolymer Chemistry in Drug Discovery
SynTech 04: Nucleic Acids Drugs Chemistry SynTech 17: Natural Product Discovery and Biosynthesis
SynTech 05: Fusion Peptide and Protein SynTech 18: Enantioselective Organocatalysis in Medichem
SynTech 06: Medichem for Better Protein Drugs SynTech 19: Continuous Flow Chemistry in Medicinal Chemistry
SynTech 07: Medichem for Antibody-Drug Conjugates SynTech 20: Medicinal Organometallic Chemistry
SynTech 08: Vaccine Medicinal Chemistry SynTech 21: Diversity-Oriented Synthesis
SynTech 09: Synthetic Biology in Medicinal Chemistry SynTech 22: Biosynthesis to Construct Complex Molecules
SynTech 10: Template Guided Systems SynTech 23: New Catalysis in Medicinal Chemistry
SynTech 11: Art of Total Synthesis SynTech 24: Isotope labeling Chemistry for Drug Discovery
SynTech 12: Carbohydrate-based Medicinal Chemistry SynTech 25: Heterocycles in Medicinal Chemistry
SynTech 13: Solid Phase and Combinatorial Chemistry SynTech 26: Structure-biodegradability Relationship

Stage 7: Accelerators of Bio/Physical Testing
-Shortening the Preclinical Process

Platform 01: Innovative Drug Screening Platform 05: Chemical, Bio/Physical Tools for Early Clinical Trials
Platform 02: HT Chemistry for Hit and Lead Synthesis Platform 06: Target Deconvolution, Validation and Target Discovery
Platform 03: Microfluidics, Mesofluidics, and Lab-on-a-chip Technologies Platform 07: Predictive Toxicology in Drug Safety
Platform 04: New Drug Discovery Screening Cascades
-In Vitro, Ex-Vivo, and In Vivo
Platform 08: Drug Efficacy Evaluation

Stage 8: Integrative Discovery Chemistry Servers
-Future of CRO, CSO, CMO, CXO

Platform 01: Discovery Process Services
-Target Selection, Validation, and Lead Optimization
Platform 05: Small Molecule Discovery Services
Platform 02: ADMEX and DMPK Services Platform 06: Clinical Trial Services
Platform 03: Medicinal Chemistry
-Drug Candidate In Vitro and In Vivo Evaluations
Platform 07: Biotherapy R & D Services
Platform 04: CMO Services of GLP and GMP Synthesis Platform 08: CMC Regulatory Affair Services

Stage 9: Smart Inventors Hackling Unmet Diseases
-Pipeline Briefing on Next $Billion Solutions to Unsolved Man’s Disorders

Hub 01: Small Molecule Immuno-Oncology Hub 09: Pain & Addiction
Hub 02: Targeting Anticancer Drugs Hub 10: Blood and Blood Organ Generation Diseases
Hub 03: Novel Cardiovascular Drugs Hub 11: Inflammatory and Immune Diseases
Hub 04: CNS Diseases and Pain Hub 12: Bone Diseases
Hub 05: GI, Liver and Disorders Hub 13: Skin Disorders
Hub 06: New Antivirals and Challenging Antibacterials
-Hackling Emerging Infections and Drug Resistance
Hub 14: Genito Urinary and Regeneration Organ Diseases
Hub 07: Anti-Aging Drugs Diabetes & Obese Hub 15: Metabolic and Hormone Disorders
Hub 08: Respiratory Diseases Hub 16: Rare Diseases

Stage 10: Futurists of Discovery Chemistry
-Young Chemists’ Short Talk and Poster Sessions

Nexus 1: Innovation in Target Discovery Nexus 4: Drug Screening and Hit-to-Lead Optimization
Nexus 2: AI/ML/DL in Medicinal Chemistry Nexus 5: Smart Drug Characterization Technology for Candidates
Nexus 3: ADMET/PKPD of Biotherapy Nexus 6: Green Medichem/Pharmaceutical Process Chemistry

Stage 11: Women Experts in Medichem
-Making Medichem World Family Diversified

Forum 01: Women Leadership in Medicinal Chemistry Forum 03: Women’s Creativity in Drug Design
Forum 02: Women’s Innovations in Medichem Forum 04: Women’s Innovative Chemistry

Stage 12: Great Mentors of New Concepts in Medichem
-Knowledge Drives to Success

Workshop 01: Chemical Biology & Medicinal Chemistry Workshop 07: Robotics and Automations in Medichem
Workshop 02: Synthetic Biology in Medichem Workshop 08: Continuous Flow Technology
Workshop 03: Quantum Chemistry in Medicinal Chemistry Workshop 09: Biomolecular Medicinal Chemistry
Workshop 04: Bimolecular Simulations Workshop 10: Small Molecules for Immuno-Oncology Therapeutics
Workshop 05: Retrometabolic Drug Design Workshop 11: Precision Medicine and Medicinal Chemistry
Workshop 06: New Virtual Reality Tool for Structure-Based Drug Design Workshop 12: New Synthetic Technologies in Medichem

Joint Conferences

Theme 1: Joint Satellite Clustering Meetings of IDDST-Macao 2021
Theme 2: Joint Satellite Clustering Meetings of SDDS-Macao 2021
Theme 3: Joint Satellite Clustering Meetings of IO-Macao 2021
Theme 4: Joint Satellite Clustering Meetings of GCC-Macao 2021
Theme 5: Joint Satellite Clustering Meetings of Synbio+-Macao 2021
S 4-1: When Entrepreneurs Meet with VCs S 4-5: Project Matchmaking
S 4-2: BP Roadshow S 4-6: PSA Onsite: 1 to 1/Face to Face Meetings
S 4-3: Industry Park Briefing S 4-7: Meet Your Future Mentors
S 4-4: New Tech/Products News Release Conference S 4-8: Talents Recruitment Fair

Posters and Exhibition

Zone 1: Poster Shows Zone 2: New Technologies and Products Exhibition

Branding Building and Cultural Activities

Activity 1: Welcome Banquet and Award Ceremony Activity 4: Field Trip to Parks
Activity 2: Industrial Sponsored Lunch Showcase and Cocktail Party Activity 5: Macao Impression Tech-Tour
Activity 3: Master Tours to Campus Activity 6: Closing and Signing Ceremony
News Updates
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