BIT's 14^th Annual Congress of International Drug Discovery Science and Technology-South Korea 2016 (IDDST-South Korea 2016), hosted by BIT Group Global Ltd., supported by Goyang City, Gyeonggi MICE Bureau and Gyeonggi Tourism Organization, was grandly held in Korea International Exhibition Center (KINTEX), Gyeonggi, South Korea on June 16^th. More than 180 specialists from 35 countries and areas attended the 3-days congress. The opening ceremony and the forum was conducted by Jianxun Xie, Director of toxicology of Shanghai Innovation Center of Roche Pharmaceuticals Ltd., and many honored guests delivered brilliant keynote speeches which last approximately three hours, among them are: Dr. Chris Senanayake, Vice President of Department of Chemical Development in Boehringer Ingelheim Pharmaceuticals, Inc.; Dr. Bruce Given, COO of Arrowhead Research Corporation; Dr. Joseph P. Thomas, Chair of the Life Sciences Group and Co-chair of the Litigation Department in Ulmer & Berne LLP; Mr. Sean Hall, CEO of Medlab Clinical Ltd.; Dr. Seonggu Ro, Executive Vice President & CTO of Crystal Genomics, Inc. …etc. This Congress comprised 20 sessions, on which more than 130 specialists gave wonderful speeches.